Number of Chains

SCOPe

[ABCDEF][a]

PDB Entries

PDB ID OPM Mutant Chain Formula Resolution HETNAM
Amino Acid sequence SCOPe Family Level CATH Homology Level
1a0r [ABC] [ABC] [ABC] 2.8
ACE:ACETYL GROUP
FAR:FARNESYL
1b9x [ABC] [ABC] [ABC] 3
GD:GADOLINIUM ATOM
1b9y [ABC] [ABC] [ABC] 3
GD:GADOLINIUM ATOM
1gg2 [ABC] [ABC] [ABC] 2.4
GDP:GUANOSINE-5___sq___-DIPHOSPHATE
1got [ABC] [ABC] [ABC] 2
GDP:GUANOSINE-5___sq___-DIPHOSPHATE
MSE:SELENOMETHIONINE
1gp2 [ABC] [ABC] [ABC] 2.3
GDP:GUANOSINE-5___sq___-DIPHOSPHATE
1omw [ABC] [ABC] [ABC] 2.5
CMT:O-METHYLCYSTEINE
1tbg [A4B4] [A4B4] [A4B4] 2.1
1xhm [AB][a] [AB][a] [AB][a] 2.7
2bcj [ABCD] [ABCD] [ABCD] 3.06
ACE:ACETYL GROUP
ALF:TETRAFLUOROALUMINATE ION
GDP:GUANOSINE-5___sq___-DIPHOSPHATE
MG:MAGNESIUM ION
2trc [ABC] [ABC] [ABC] 2.4
GD:GADOLINIUM ATOM
MSE:SELENOMETHIONINE
3ah8 [ABC][a] [ABC][a] [ABC][a] 2.9
ACE:ACETYL GROUP
DAM:N-METHYL-ALPHA-BETA-DEHYDROALANINE
GDP:GUANOSINE-5___sq___-DIPHOSPHATE
HF2:(2R)-2-HYDROXY-3-PHENYLPROPANOIC ACID
HL2:(2S,3R)-2-AMINO-3-HYDROXY-4-METHYLPENTANOIC ACID
MAA:N-METHYL-L-ALANINE
OTH:N,O-DIMETHYL-L-THREONINE
THC:N-METHYLCARBONYLTHREONINE
3cik [ABC] [ABC] [ABC] 2.75
CMT:O-METHYLCYSTEINE
MG:MAGNESIUM ION
3krw [ABC] [ABC] [ABC] 2.9
BA1:BALANOL
CMT:O-METHYLCYSTEINE
MG:MAGNESIUM ION
3krx [ABC] [ABC] [ABC] 3.1
BA1:BALANOL
CMT:O-METHYLCYSTEINE
MG:MAGNESIUM ION
3psc [ABC] [ABC] [ABC] 2.67
CMT:O-METHYLCYSTEINE
3pvu [ABC] [ABC] [ABC] 2.48
CMT:O-METHYLCYSTEINE
QRW:3-({[4-METHYL-5-(PYRIDIN-4-YL)-4H-1,2,4-TRIAZOL-3-YL]METHYL}AMINO)-N-[2-(TRIFLUOROMETHYL)BENZYL]BENZAMIDE
3pvw [ABC] [ABC] [ABC] 2.49
CMT:O-METHYLCYSTEINE
QRX:N-(2,6-DIFLUOROBENZYL)-3-({[4-PROPYL-5-(PYRIMIDIN-4-YL)-4H-1,2,4-TRIAZOL-3-YL]METHYL}AMINO)BENZAMIDE
3v5w [ABC] [ABC] [ABC] 2.07
8PR:PAROXETINE
MG:MAGNESIUM ION
4pnk [ABC] [ABC] [ABC] 2.56
KZQ:(4S)-4-(4-FLUOROPHENYL)-N-(2H-INDAZOL-5-YL)-6-METHYL-2-OXO-1,2,3,4-TETRAHYDROPYRIMIDINE-5-CARBOXAMIDE
5he0 [ABC] [ABC] [ABC] 2.56
453:(4S)-4-{4-FLUORO-3-[(PYRIDIN-2-YLMETHYL)CARBAMOYL]PHENYL}-N-(1H-INDAZOL-5-YL)-6-METHYL-2-OXO-1,2,3,4-TETRAHYDROPYRIMIDINE-5-CARBOXAMIDE
5he1 [ABC] [ABC] [ABC] 3.15
MG:MAGNESIUM ION
ZS2:(4~{S})-4-[4-FLUORANYL-3-(ISOQUINOLIN-1-YLMETHYLCARBAMOYL)PHENYL]-~{N}-(1~{H}-INDAZOL-5-YL)-6-METHYL-2-OXIDANYLIDENE-3,4-DIHYDRO-1~{H}-PYRIMIDINE-5-CARBOXAMIDE
5he2 [ABC] [ABC] [ABC] 2.79
F0S:(4~{S})-4-[3-[(2,6-DIMETHOXYPHENYL)METHYLCARBAMOYL]-4-FLUORANYL-PHENYL]-~{N}-(1~{H}-INDAZOL-5-YL)-6-METHYL-2-OXIDANYLIDENE-3,4-DIHYDRO-1~{H}-PYRIMIDINE-5-CARBOXAMIDE
5he3 [ABC] [ABC] [ABC] 2.74
FF1:(4~{S})-4-[3-[2-(2,6-DIMETHYLPHENYL)ETHYLCARBAMOYL]-4-FLUORANYL-PHENYL]-~{N}-(1~{H}-INDAZOL-5-YL)-6-METHYL-2-OXIDANYLIDENE-3,4-DIHYDRO-1~{H}-PYRIMIDINE-5-CARBOXAMIDE
MG:MAGNESIUM ION
5tdh [ABC] [ABC] [ABC] 3
GDP:GUANOSINE-5___sq___-DIPHOSPHATE
5ukk [ABC] [ABC] [ABC] 2.6
8DJ:5-[(3S,4R)-3-{[(2H-1,3-BENZODIOXOL-5-YL)OXY]METHYL}PIPERIDIN-4-YL]-2-FLUORO-N-[(PYRIDIN-2-YL)METHYL]BENZAMIDE
MG:MAGNESIUM ION
5ukl [ABC] [ABC] [ABC] 2.15
MG:MAGNESIUM ION
SIX:2-{5-[(3S,4R)-3-{[(2H-1,3-BENZODIOXOL-5-YL)OXY]METHYL}PIPERIDIN-4-YL]-2-FLUOROPHENYL}-N-[2-(1H-PYRAZOL-4-YL)ETHYL]ACETAMIDE
5ukm [ABC] [ABC] [ABC] 3.03
CMT:O-METHYLCYSTEINE
MG:MAGNESIUM ION
T0E:5-[(3S,4R)-3-{[(2H-1,3-BENZODIOXOL-5-YL)OXY]METHYL}PIPERIDIN-4-YL]-2-FLUORO-N-[(1H-PYRAZOL-5-YL)METHYL]BENZAMIDE
5wg3 [ABC] [ABC] [ABC] 2.9
AFM:2-FLUORO-5-[(3S,4R)-3-{[(1H-INDAZOL-5-YL)OXY]METHYL}PIPERIDIN-4-YL]-N-[(1H-PYRAZOL-3-YL)METHYL]BENZAMIDE
MG:MAGNESIUM ION
5wg4 [ABC] [ABC] [ABC] 2.31
AFV:2-FLUORO-5-[(3S,4R)-3-{[(1H-INDAZOL-5-YL)OXY]METHYL}PIPERIDIN-4-YL]-N-[(PYRIDIN-2-YL)METHYL]BENZAMIDE
5wg5 [ABC] [ABC] [ABC] 3.1
MG:MAGNESIUM ION
ZSO:5-{[(3S,4R)-4-(4-FLUOROPHENYL)PIPERIDIN-3-YL]METHOXY}-2H-INDAZOLE
6c2y [ABC] [ABC] [ABC] 2.74
EJS:(4R,5R,6S)-4-[4-FLUORO-3-({[3-(METHOXYMETHYL)-1,2,4-OXADIAZOL-5-YL]METHYL}CARBAMOYL)PHENYL]-N-(2H-INDAZOL-5-YL)-6-METHYL-2-OXOHEXAHYDROPYRIMIDINE-5-CARBOXAMIDE
6crk [ABCD] [ABCD] [ABCD] 2
FLC:CITRATE ANION
GDP:GUANOSINE-5___sq___-DIPHOSPHATE
6eg8 [ABC] [ABC] [ABC] 2.8
GDP:GUANOSINE-5___sq___-DIPHOSPHATE
MG:MAGNESIUM ION
6k41 [ABCDE] [ABCDE] [ABCDE] ELECTRON MICROSCOPY
2.9
CZX:4-[(1~{S})-1-(2,3-DIMETHYLPHENYL)ETHYL]-1~{H}-IMIDAZOLE
6kpf [ABCDE] [ABCDE] [ABCDE] ELECTRON MICROSCOPY
2.9
E3R:7-[(6AR,9R,10AR)-1-HYDROXY-9-(HYDROXYMETHYL)-6,6-DIMETHYL-6A,7,8,9,10,10A-HEXAHYDRO-6H-BENZO[C]CHROMEN-3-YL]- 7-METHYLOCTANENITRILE
6kpg [ABCDE] [ABCDE] [ABCDE] ELECTRON MICROSCOPY
3
8D0:(6~{A}~{R},9~{R},10~{A}~{R})-9-(HYDROXYMETHYL)-3-(8-ISOTHIOCYANATO-2-METHYL-OCTAN-2-YL)-6,6-DIMETHYL-6~{A},7,8,9,10,10~{A}-HEXAHYDROBENZO[C]CHROMEN-1-OL
6n4b [ABCDE] [ABCDE] [ABCDE] ELECTRON MICROSCOPY
3
CLR:CHOLESTEROL
KCA:METHYL N-{1-[(4-FLUOROPHENYL)METHYL]-1H-INDAZOLE-3-CARBONYL}-3-METHYL-L-VALINATE
6u7c [ABC] [ABC] [ABC] 2.44
MG:MAGNESIUM ION
Q1Y:5-[(3S,4R)-3-{[(2H-1,3-BENZODIOXOL-5-YL)OXY]METHYL}PIPERIDIN-4-YL]-2-FLUORO-N-[(2H-INDAZOL-3-YL)METHYL]BENZAMIDE
6x19 [ABCDE] [ABCDE] [ABCDE] ELECTRON MICROSCOPY
2.1
UK1:3-{(1S)-1-[5-(2,2-DIMETHYLMORPHOLIN-4-YL)-2-{(4S)-2-(4-FLUORO-3,5-DIMETHYLPHENYL)-3-[3-(4-FLUORO-1-METHYL-1H-INDAZOL-5-YL)-2-OXO-2,3-DIHYDRO-1H-IMIDAZOL-1-YL]-4-METHYL-2,4,6,7-TETRAHYDRO-5H-PYRAZOLO[4,3-C]PYRIDINE-5-CARBONYL}-1H-INDOL-1-YL]BUTYL}-1,2,4-OXADIAZOL-5(4H)-ONE
6x1a [ABCDE] [ABCDE] [ABCDE] ELECTRON MICROSCOPY
2.5
UK4:2-[(4-{6-[(4-CYANO-2-FLUOROPHENYL)METHOXY]PYRIDIN-2-YL}PIPERIDIN-1-YL)METHYL]-1-{[(2S)-OXETAN-2-YL]METHYL}-1H-BENZIMIDAZOLE-6-CARBOXYLIC ACID
6xbm [ABCDE] [ABCDE] [ABCDE] ELECTRON MICROSCOPY
3.15
CO1:17-[3-(3,3-DIMETHYL-OXIRANYL)-1-METHYL-PROPYL]-10,13-DIMETHYL-2,3,4,7,8,9,10,11,12,13,14,15,16,17-TETRADECAHYDRO-1H-CYC LOPENTA[A]PHENANTHREN-3-OL
6xox [ABCDEF] [ABCDEF] [ABCDEF] ELECTRON MICROSCOPY
3.1
V6G:3-[(1S,2S)-1-(5-[(4S)-2,2-DIMETHYLOXAN-4-YL]-2-{(4S)-2-(4-FLUORO-3,5-DIMETHYLPHENYL)-3-[3-(4-FLUORO-1-METHYL-1H-INDAZOL-5-YL)-2-OXO-2,3-DIHYDRO-1H-IMIDAZOL-1-YL]-4-METHYL-2,4,6,7-TETRAHYDRO-5H-PYRAZOLO[4,3-C]PYRIDINE-5-CARBONYL}-1H-INDOL-1-YL)-2-METHYLCYCLOPROPYL]-1,2,4-OXADIAZOL-5(4H)-ONE
7ckz [ABCDE] [ABCDE] [ABCDE] ELECTRON MICROSCOPY
3.1
CLR:CHOLESTEROL
G4C:2-[2,6-BIS(CHLORANYL)PHENYL]-1-[(1S,3R)-3-(HYDROXYMETHYL)-1-METHYL-5-(3-METHYL-3-OXIDANYL-BUTYL)-3,4-DIHYDRO-1H-ISOQUINOLIN-2-YL]ETHANONE
LDP:L-DOPAMINE
7cmu [ABCDE] [ABCDE] [ABCDE] ELECTRON MICROSCOPY
3
G6L:(6S)-N6-PROPYL-4,5,6,7-TETRAHYDRO-1,3-BENZOTHIAZOLE-2,6-DIAMINE
7cmv [ABCDE] [ABCDE] [ABCDE] ELECTRON MICROSCOPY
2.7
G6O:(4AR,10BR)-4-PROPYL-3,4A,5,10B-TETRAHYDRO-2H-CHROMENO[4,3-B][1,4]OXAZIN-9-OL
7d76 [ABCD] [ABCD] [ABCD] ELECTRON MICROSCOPY
3.1
CLR:CHOLESTEROL
GXR:(8~{S},9~{R},10~{S},11~{S},13~{S},14~{S},16~{S},17~{R})-9-CHLORANYL-10,13,16-TRIMETHYL-11,17-BIS(OXIDANYL)-17-(2-OXIDANYLETHANOYL)-6,7,8,11,12,14,15,16-OCTAHYDROCYCLOPENTA[A]PHENANTHREN-3-ONE
PLM:PALMITIC ACID
Y01:CHOLESTEROL HEMISUCCINATE
7e32 [ABCDE] [ABCDE] [ABCDE] ELECTRON MICROSCOPY
2.9
CLR:CHOLESTEROL
SRO:SEROTONIN
7e33 [ABCDE] [ABCDE] [ABCDE] ELECTRON MICROSCOPY
2.9
HVU:3-(1-METHYLPIPERIDIN-4-YL)-1H-INDOL-5-OL
7f1q [ABCD] [ABCD] [ABCD] ELECTRON MICROSCOPY
2.9
7f1r [ABCD] [ABCD] [ABCD] ELECTRON MICROSCOPY
3
7f1s [ABCD] [ABCD] [ABCD] ELECTRON MICROSCOPY
2.8
7jjo [ABCDE] [ABCDE] [ABCDE] ELECTRON MICROSCOPY
2.6
5FW:ISOPRENALINE
7k7l [ABC] [ABC] [ABC] 2.54
MG:MAGNESIUM ION
W4D:3-BENZYL-6-(1H-PYRAZOL-4-YL)QUINAZOLIN-4(3H)-ONE
7k7z [ABC] [ABC] [ABC] 2.61
W4G:3-BENZYL-7-(1H-PYRAZOL-4-YL)QUINAZOLIN-4(3H)-ONE
7kh0 [ABCDEF][a] [ABCDEF][a] [ABCDEF][a] ELECTRON MICROSCOPY
2.8
NH2:AMINO GROUP
7l1v [ABCDEF] [ABCDEF] [ABCDEF] ELECTRON MICROSCOPY
3
XGD:4___sq___-METHOXY-N,N-DIMETHYL-3___sq___-{[3-(2-{[2-(2H-1,2,3-TRIAZOL-2-YL)BENZENE-1-CARBONYL]AMINO}ETHYL)PHENYL]SULFAMOYL}[1,1___sq___-BIPHENYL]-3-CARBOXAMIDE
7lci [ABCD] [ABCD] [ABCD] ELECTRON MICROSCOPY
2.9
UK4:2-[(4-{6-[(4-CYANO-2-FLUOROPHENYL)METHOXY]PYRIDIN-2-YL}PIPERIDIN-1-YL)METHYL]-1-{[(2S)-OXETAN-2-YL]METHYL}-1H-BENZIMIDAZOLE-6-CARBOXYLIC ACID
7ljc [ABCDE] [ABCDE] [ABCDE] ELECTRON MICROSCOPY
3
CLR:CHOLESTEROL
G4C:2-[2,6-BIS(CHLORANYL)PHENYL]-1-[(1S,3R)-3-(HYDROXYMETHYL)-1-METHYL-5-(3-METHYL-3-OXIDANYL-BUTYL)-3,4-DIHYDRO-1H-ISOQUINOLIN-2-YL]ETHANONE
PLM:PALMITIC ACID
SK0:(1R)-6-CHLORO-1-PHENYL-2,3,4,5-TETRAHYDRO-1H-3-BENZAZEPINE-7,8-DIOL
*Chain Formula of OLIGAMI.
  [ ] : Polypeptide - [AB] : Protein, [ab] : Small peptide
  ( ) : Nucleic acid - (AB) : DNA, (ab) : RNA
PDL